4pvo A 1.48 BS03 S3C A 1 W87 H118 D120 H196 C221 N233 H263 W56 H85 D87 H148 C167 N179 H209 H116 H118 D120 H196 C221 Y224 N233 H263 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0046872 Q9K2N0 25411887 403 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 4pvo B 1.48 BS03 S3C B 1 W87 H118 D120 H196 C221 N233 H263 W56 H85 D87 H148 C167 N179 H209 H116 H118 D120 H196 C221 Y224 N233 H263 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0046872 Q9K2N0 25411887 406 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNRSV 4pvt A 2.0 BS03 S3C A 1 W87 H118 D120 H196 C221 N233 H263 W56 H85 D87 H148 C167 N179 H209 H116 H118 D120 H196 C221 Y224 N233 H263 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0046872 -logKd/Ki=6.52, IC50=0.3uM Q9K2N0 25411887 403 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 4pvt B 2.0 BS03 S3C B 1 W87 H118 D120 H196 C221 N233 H263 W56 H85 D87 H148 C167 N179 H209 H116 H118 D120 H196 C221 Y224 N233 H263 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0046872 Q9K2N0 25411887 406 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 4tyt A 1.799 BS03 S3C A 1 W89 H118 D120 H179 C198 N210 H240 W50 H79 D81 H140 C159 N171 H201 H116 H118 D120 H179 C198 K201 N210 H240 H77 H79 D81 H140 C159 K162 N171 H201 3.5.2.6 0008270,0008800,0016787,0017001,0042597,0046677,0046872 ic50=0.02uM -logKd/Ki=7.70, IC50=0.02uM IC50=80nM P04190 25411887 303 EKTVIKNTGTISISQLNKNVWVHTELGSAVPSNGLVLNTSKGLVLVDSSWDDKLTKELIEMVEKKFQKRVTDVIITHAHADRIGGIKTLKERGIKAHSTALTAELAKKNGYEEPLGDLQTVTNLKFGNMKVETFYPGKGHTEDNIVVWLPQYNILVGGCLVKSTSAKDLGNVADAYVNEWSTSIENVLKRYRNINAVVPGHGEVGDKGLLLHTLDLLK 5n5h A 1.3 BS03 S3C A 1 F62 W87 H116 D118 H179 C198 N210 H240 F32 W57 H86 D88 H149 C168 N180 H210 H114 H116 D118 H179 C198 H201 N210 H240 H84 H86 D88 H149 C168 H171 N180 H210 3.5.2.6 0016787,0017001,0046872 Q9XAY4 30430727 303 GEYPTVNEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEAEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSANVLYGGCAVHELSSTSAGNVADADLAEWPTSVERIQKHYPEAEVVIPGHGLPGGLDLLQHTANVVKAHKNRSV 6ew3 A 2.14 BS03 S3C A 1 W87 H116 D118 H179 C198 N210 H240 W56 H85 D87 H148 C167 N179 H209 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0046872 ic50=0.04uM -logKd/Ki=7.40, IC50=0.04uM D1MEN9 29655609 506 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR 6ew3 B 2.14 BS03 S3C B 1 W87 H116 D118 H179 C198 N210 H240 W56 H85 D87 H148 C167 N179 H209 H114 H116 D118 H179 C198 Y201 N210 H240 H83 H85 D87 H148 C167 Y170 N179 H209 3.5.2.6 0016787,0017001,0046872 ic50=0.04uM D1MEN9 29655609 506 EYPTVSEIPVGEVRLYQIADGVWSHIATQSFDGAVYPSNGLIVRDGDELLLIDTAWGAKNTAALLAEIEKQIGLPVTRAVSTHFHDDRVGGVDVLRAAGVATYASPSTRRLAEVEGNEIPTHSLEGLSSSGDAVRFGPVELFYPGAAHSTDNLVVYVPSASVLYGGCAIYELSRTSAGNVADADLAEWPTSIERIQQHYPEAQFVIPGHGLPGGLDLLKHTTNVVKAHTNR