2fm5 A 2.03 BS02 M99 A 1 M273 D318 N321 Y329 W332 T333 I336 M357 Q369 F372 M195 D240 N243 Y251 W254 T255 I258 M279 Q291 F294 3.1.4.53 0004114,0007165,0008081 ic50=43nM -logKd/Ki=7.37, IC50=43nM IC50=43nM Q08499 16539372 601 IPRFGVKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPQ 2fm5 B 2.03 BS02 M99 B 1 M273 D318 N321 P322 W332 T333 I336 M357 Q369 F372 M188 D233 N236 P237 W247 T248 I251 M272 Q284 F287 3.1.4.53 0004114,0007165,0008081 ic50=43nM IC50=43nM Q08499 16539372 602 TEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPQ 2fm5 C 2.03 BS02 M99 C 1 M273 D318 N321 P322 Y329 W332 T333 I336 M357 Q369 F372 M188 D233 N236 P237 Y244 W247 T248 I251 M272 Q284 F287 3.1.4.53 0004114,0007165,0008081 ic50=43nM IC50=43nM Q08499 16539372 603 TEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPQ 2fm5 D 2.03 BS02 M99 D 1 M273 D318 N321 P322 Y329 W332 T333 I336 M357 Q369 F372 M195 D240 N243 P244 Y251 W254 T255 I258 M279 Q291 F294 3.1.4.53 0004114,0007165,0008081 ic50=43nM IC50=43nM Q08499 16539372 604 IPRFGVKTEQEDVLAKELEDVNKWGLHVFRIAELSGNRPLTVIMHTIFQERDLLKTFKIPVDTLITYLMTLEDHYHADVAYHNNIHAADVVQSTHVLLSTPALEAVFTDLEILAAIFASAIHDVDHPGVSNQFLINTNSELALMYNDSSVLENHHLAVGFKLLQEENCDIFQNLTKKQRQSLRKMVIDIVLATDMSKHMNLLADLKTMVETKKVTSSGVLLLDNYSDRIQVLQNMVHCADLSNPTKPLQLYRQWTDRIMEEFFRQGDRERERGMEISPMCDKHNASVEKSQVGFIDYIVHPLWETWADLVHPDAQDILDTLEDNREWYQSTIPQ