6mdd A 2.05 BS01 JE7 A 1 R111 T218 T219 E250 T253 L254 P491 K492 Q495 R101 T199 T200 E221 T224 L225 P443 K444 Q447 D425 C459 R465 T466 Q506 D377 C411 R417 T418 Q458 3.1.3.48 0004725,0006470,0016311 ic50=47uM -logKd/Ki=4.33, IC50=47uM Q06124 30688462 601 SRRWFHPNITGVEAENLLLTRGVDGSFLARPSKSNPGDFTLSVRRNGAVTHIKIQNTGDYYDLYGGEKFATLAELVQYYMEHGDVIELKYPLNCADPTSERWFHGHLSGKEAEKLLTEKGKHGSFLVRESQSHPGDFVLSVRTGDSKVTHVMIRCQELKYDVGGGERFDSLTDLVEHYKKNPMVETLGTVLQLKQPLNTTRINAAEIESRVRELSKGFWEEFETLQQQECKLLYSRKEGQRQENKNKNRYKNILPFDHTRVVLHDSDYINANIIMPKSYIATQGCLQNTVNDFWRMVFQENSRVIVMTTKEVERGKSKCVKYWPDEYALKEYGVMRVRNVKESAAHDYTLRELKLSKVGQGNTERTVWQYHFRTWPDHGVPSDPGGVLDFLEEVHHKQESIMDAGPVVVHCSAGIGRTGTFIVIDILIDIIREKGVDCDIDVPKTIQMVRSQRSGMVQTEAQYRFIYMAVQHYIETL 6mdd B 2.05 BS01 JE7 B 1 R111 T218 T219 E250 T253 L254 Q257 P491 K492 Q495 R100 T193 T194 E215 T218 L219 Q222 P437 K438 Q441 D425 C459 R465 T466 Q506 D371 C405 R411 T412 Q452 3.1.3.48 0004725,0006470,0016311 ic50=47uM Q06124 30688462 601 RRWFHPNITGVEAENLLLTRGVDGSFLARPSKSNPGDFTLSVRRNGAVTHIKIQNTGDYYDLYGGEKFATLAELVQYYMEQLKVIELKYPLNCADPTSERWFHGHLSGKEAEKLLTEKGKHGSFLVREHPGDFVLSVRTSKVTHVMIRCQELKYDVGGGERFDSLTDLVEHYKKNPMVETLGTVLQLKQPLNTTRINAAEIESRVRELSKGFWEEFETLQQQECKLLYSRKEGQRQENKNKNRYKNILPFDHTRVVLHVSDYINANIIMPKSYIATQGCLQNTVNDFWRMVFQENSRVIVMTTKEVERGKSKCVKYWPDEYALKEYGVMRVRNVKESAAHDYTLRELKLSKVGQGNTERTVWQYHFRTWPDHGVPSDPGGVLDFLEEVHHKQESIMDAGPVVVHCSAGIGRTGTFIVIDILIDIIREKGVDCDIDVPKTIQMVRSQRSGMVQTEAQYRFIYMAVQHYIETL