2csn A 2.5 BS01 CKI A 1 I18 I26 L88 L138 I13 I21 L83 L133 2.7.11.1 0004672,0005524,0006468 Ki=39uM -logKd/Ki=4.41, Ki=39uM P40233 8692811 300 NVVGVHYKVGRRIGEGSFGVIFEGTNLLNNQQVAIKFEPRRSDAPQLRDEYRTYKLLAGCTGIPNVYYFGQEGLHNVLVIDLLGPSLEDLLDLCGRKFSVKTVAMAAKQMLARVQSIHEKSLVYRDIKPDNFLIGRPNSKNANMIYVVDFGMVKFYRDPVTKQHIPYREKKNLSGTARYMSINTHLGREQSRRDDLEALGHVFMYFLRGSLPWQGLKAATNKQKYERIGEKKQSTPLRELCAGFPEEFYKYMHYARNLAFDATPDYDYLQGLFSKVLERLNTTEDENFDWNLL 3q2j A 2.1501 BS02 CKI A 1 M26 Y42 M90 E92 A93 L97 S194 F197 I207 M23 Y39 M87 E89 A90 L94 S191 F194 I204 K44 D190 N195 D208 K41 D187 N192 D205 2.7.1.95 0005524,0008910,0016301,0016310,0016773,0046677 -logKd/Ki=4.18, Ki=66.1uM P0A3Y5 21573013 300 MRISPELKKLIEKYRCVKDTEGMSPAKVYKLVGENENLYLKMTDSRYKGTTYDVEREKDMMLWLEGKLPVPKVLHFERHDGWSNLLMSEADGVLCSEEYEDEQSPEKIIELYAECIRLFHSIDISDCPYTNSLDSRLAELDYLLNNDLADVDCENWEEDTPFKDPRELYDFLKTEKPEEELVFSHGDLGDSNIFVKDGKVSGFIDLGRSGRADKWYDIAFCVRSIREDIGEEQYVELFFDLLGIKPDWEKIKYYILLDELF 3q2j B 2.1501 BS02 CKI B 1 Y42 M90 A93 L97 S194 F197 I207 Y41 M89 A92 L96 S193 F196 I206 K44 D190 N195 D208 K43 D189 N194 D207 2.7.1.95 0005524,0008910,0016301,0016310,0016773,0046677 P0A3Y5 21573013 300 AKMRISPELKKLIEKYRCVKDTEGMSPAKVYKLVGENENLYLKMTDSRYKGTTYDVEREKDMMLWLEGKLPVPKVLHFERHDGWSNLLMSEADGVLCSEEYEDEQSPEKIIELYAECIRLFHSIDISDCPYTNSLDSRLAELDYLLNNDLADVDCENWEEDTPFKDPRELYDFLKTEKPEEELVFSHGDLGDSNIFVKDGKVSGFIDLGRSGRADKWYDIAFCVRSIREDIGEEQYVELFFDLLGIKPDWEKIKYYILLDELF 3q2m A 2.9 BS01 CKI A 1 F50 F102 I103 A105 F48 F100 I101 A103 ? 0000166,0016740,0046872 -logKd/Ki=3.80, Ki=159uM O06916 21573013 400 KQPIQAQQLIELLKVHYGIDIHTAQFIQGGADTNAFAYQADSESKSYFIKLKYGYHDEINLSIIRLLHDSGIKEIIFPIHTLEAKLFQQLKHFKIIAYPFIHAPNGFTQNLTGKQWKQLGKVLRQIHETSVPISIQQQLRKEIYSPKWREIVRSFYNQIEFDNSDDKLTAAFKSFFNQNSAAIHRLVDTSEKLSKKIQPDLDKYVLCHSDIHAGNVLVGNEESIYIIDWDEPMLAPKERDLMFIGGGVGNVWNKPHEIQYFYEGYGEINVDKTILSYYRHERIVEDIAVYGQDLLSRNQNNQSRLESFKYFKEMFDPNNVVEIAFATEQ 4xhl A 3.01 BS01 CKI A 1 I15 I23 A36 L85 D91 L135 I148 I11 I14 A27 L76 D82 L126 I139 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=4.43, IC50=37uM P29295 27491543 401 VGRKFRIGRKIGDIYHGTNLISGEEVAIRLESIRSRHPQLDYESRVYRYLSGGVGIPFIRWFGREGEYNAMVIDLLGPSLEDLFNYCHRRFSFKTVIMLALQMFCRIQYIHGRSFIHRDIKPDNFLMGVGRRGSTVHVIDFGLSKKYRDFNTHRHIPYRENKSLTGTARYASVNTHLGIEQSRRDDLESLGYVLIYFCKGSLPWQGLKATTKKQKYDRIMEKKLNVSVETLCSGLPLEFQEYMAYCKNLKFDEKPDYLFLARLFKDLSIKLEYHNDHLFDWTMLRYTKAMTFNKIKLLAMKKFPTHFHYYKNEDKHNPSPEEIKQQTILN