3v8t A 2.0 BS01 477 A 1 I369 A389 K391 F435 E436 F437 M438 H440 G441 L489 I15 A32 K34 F78 E79 F80 M81 H83 G84 L132 D482 A484 R486 N487 D500 P521 D125 A127 R129 N130 D143 P147 2.7.10.2 0004672,0004713,0004715,0005524,0006468 ic50=0.3nM -logKd/Ki=9.52, IC50=0.3nM Q08881 22464456 701 GSVIDPSELTFVQEIGSGLVHLGYWLNKDKVAIKTIREGAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAES 3v8t B 2.0 BS01 477 B 1 I369 A389 K391 F435 E436 F437 M438 G441 L489 I15 A33 K35 F76 E77 F78 M79 G82 L130 D482 A484 R486 N487 D500 P521 D123 A125 R127 N128 D141 P146 2.7.10.2 0004672,0004713,0004715,0005524,0006468 ic50=0.3nM Q08881 22464456 701 GSVIDPSELTFVQEIGSGGLVHLGYWLNKDKVAIKTIAMSEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAESG 3vf9 A 2.3 BS01 477 A 1 L377 A400 M448 E449 M450 A451 L453 G454 P455 L501 L14 A36 M78 E79 M80 A81 L83 G84 P85 L131 D494 A496 R498 N499 D512 K533 D124 A126 R128 N129 D142 K163 2.7.10.2 0004672,0004713,0005524,0006468 ic50=358.2nM -logKd/Ki=8.72, IC50=1.9nM P43405 22464456 701 YLDRKLLTLEDKELGSGNFGTVKKGYYQMKVVKTVAVKILPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVN